
Azasetron hydrochloride
CAS No. 123040-16-4
Azasetron hydrochloride( Azasetron hydrochloride | Y 25130 | Y-25130 | Y25130. )
Catalog No. M10908 CAS No. 123040-16-4
Azasetron Hydrochloride is a 5-HT3 receptor antagonist which is used as an anti-emetic.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
5MG | 31 | In Stock |
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10MG | 48 | In Stock |
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25MG | 86 | In Stock |
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50MG | 157 | In Stock |
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100MG | 266 | In Stock |
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200MG | Get Quote | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameAzasetron hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionAzasetron Hydrochloride is a 5-HT3 receptor antagonist which is used as an anti-emetic.
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DescriptionAzasetron Hydrochloride is a 5-HT3 receptor antagonist which is used as an anti-emetic.Azasetron inhibited the specific binding of [3H]quipazine to 5-HT3 receptors at the synaptic membranes of the rat cerebral cortex.(In Vivo):Azasetron could effectively penetrate through the skin and pass into the systemic circulation.
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In Vitro——
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In VivoAzasetron could effectively penetrate through the skin and pass into the systemic circulation. Animal Model:Four male Bama miniature pigs weighing 9-11 kg (15-16 weeks old).Dosage:0.5 mg/kg.Administration:I.V. administration via the abdominal vein.Result:The mean plasma concentration dropped to minimum at 36 h. Cmax = 44.88 ± 7.16 ng/mL) was achieved at the time point of 66.00 ± 22.98 h (Tmax).
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SynonymsAzasetron hydrochloride | Y 25130 | Y-25130 | Y25130.
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT3
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Research AreaNeurological Disease
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Indication——
Chemical Information
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CAS Number123040-16-4
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Formula Weight386.27
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Molecular FormulaC17H20ClN3O3·HCl
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Purity>98% (HPLC)
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SolubilityWater: 3 mg/mL (7.76 mM)
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SMILESc1(cc(C(N[C@@H]2CN3CCC2CC3)=O)c2c(c1)N(C)C(=O)CO2)Cl.Cl
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Chemical Name2H-1,4-Benzoxazine-8-carboxamide, 3,4-dihydro-N-1-azabicyclo(2.2.2)oct-3-yl-6-chloro-4-methyl-3-oxo-, monohydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Katayama K, et al. Jpn J Pharmacol. 1997 Apr;73(4):357-60.
molnova catalog



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